Design, synthesis, in vitro, and in vivo characterization of phenylpiperazines and pyridinylpiperazines as potent and selective antagonists of the melanocortin-4 receptor

Joe A. Tran, Wanlong Jiang, Fabio C. Tucci, Beth A. Fleck, Jenny Wen, Yang Sai, Ajay Madan, Kung Chen Ta, Stacy Markison, Alan C. Foster, Sam R. Hoare, Daniel Marks, John Harman, Caroline W. Chen, Melissa Arellano, Dragan Marinkovic, Haig Bozigian, John Saunders, Chen Chen

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