Abstract
A novel class of phenylpyrazole fused Wieland-Miescher ketone derivatives are high affinity, receptor specific, selective modulators of glucocorticoid receptor (GR) function.
| Original language | English (US) |
|---|---|
| Pages (from-to) | 5199-5203 |
| Number of pages | 5 |
| Journal | Bioorganic and Medicinal Chemistry Letters |
| Volume | 14 |
| Issue number | 20 |
| DOIs | |
| State | Published - Oct 18 2004 |
| Externally published | Yes |
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Keywords
- Glucocorticoid
- Ligand
- Nuclear receptor
ASJC Scopus subject areas
- Biochemistry
- Molecular Biology
- Organic Chemistry
- Drug Discovery
- Pharmaceutical Science
Cite this
Design and evaluation of novel nonsteroidal dissociating glucocorticoid receptor ligands. / Shah, Nilesh; Scanlan, Thomas (Tom).
In: Bioorganic and Medicinal Chemistry Letters, Vol. 14, No. 20, 18.10.2004, p. 5199-5203.Research output: Contribution to journal › Article
}
TY - JOUR
T1 - Design and evaluation of novel nonsteroidal dissociating glucocorticoid receptor ligands
AU - Shah, Nilesh
AU - Scanlan, Thomas (Tom)
PY - 2004/10/18
Y1 - 2004/10/18
N2 - A novel class of phenylpyrazole fused Wieland-Miescher ketone derivatives are high affinity, receptor specific, selective modulators of glucocorticoid receptor (GR) function.
AB - A novel class of phenylpyrazole fused Wieland-Miescher ketone derivatives are high affinity, receptor specific, selective modulators of glucocorticoid receptor (GR) function.
KW - Glucocorticoid
KW - Ligand
KW - Nuclear receptor
UR - http://www.scopus.com/inward/record.url?scp=4544343929&partnerID=8YFLogxK
UR - http://www.scopus.com/inward/citedby.url?scp=4544343929&partnerID=8YFLogxK
U2 - 10.1016/j.bmcl.2004.07.052
DO - 10.1016/j.bmcl.2004.07.052
M3 - Article
C2 - 15380227
AN - SCOPUS:4544343929
VL - 14
SP - 5199
EP - 5203
JO - Bioorganic and Medicinal Chemistry Letters
JF - Bioorganic and Medicinal Chemistry Letters
SN - 0960-894X
IS - 20
ER -